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erythromycin (Erymin / erythromycin, Elan)

✓ Approved

Takeda · 小分子 · 小分子

什么是 erythromycin?

erythromycin 是一种小分子,由Takeda研发。该药已获批,用于治疗相关适应症,给药途径:Oral (PO)。

药物档案

商品名Erymin, erythromycin, Elan
公司Takeda
药物类别小分子
给药途径Oral (PO)
状态Approved

治疗适应症

erythromycin 针对 1 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Infections and infestationsSalmonellosis✓ Approved

相关研究文献

PubMedJournal of thoracic disease2026-09-11

Erythromycin inhibits the differentiation of NCR-ILC3s activated by lung dendritic cells in mice exposed to cigarette smoke.

Xu Yifang Y, Shen Ying Y, Mo Lili L, Tang Haijuan H et al.

Both dendritic cells (DCs) and nature cytotoxicity receptor-negative 3-type innate lymphoid cells (NCR-ILC3s) have been implicated in chronic lung inflammation in mice with cigarette smoke (CS)-induced chronic obstructive pulmonary disease (COPD). Our study aims to investigate whether erythromycin (EM) can suppress the differentiation of ILC3s into NCR-ILC3s through restraining DCs activation and therefore attenuate CS-related lung injuries in COPD mice. Our study comprised both in vivo and in vitro experiments. In the former, lung samples were collected from non-smokers, smokers, patients with stable COPD, as well as mice exposed to air, CS, and CS combined with EM, respectively. In the latter, lung DCs sifted by CD11c magnetic beads from mice exposed to either air or CS were co-cultured with lung CD45+Lin-CD127+ILCs sorted from air-exposed mice. EM was added to the co-culture involving DCs from CS-exposed mice. Flow cytometry and other assays were used to examine the quantities of NCR-ILC3s, DCs, relevant costimulatory molecules and cytokines in human tissues, mice lungs, and cell cultures. Compared to non-smokers, lung NCR-ILC3s frequencies significantly increased in both smokers and COPD patients, and inversely correlated with forced expiratory volume in 1 second percent predicted (FEV1% pred) and diffusing capacity for carbon monoxide (P<0.05). CS-exposed mice showed evident emphysema and elevated frequencies of lung NCR-ILC3s and DCs. In contrast, mice receiving CS and EM displayed attenuated emphysema and reduced levels of NCR-ILC3s and DCs (P<0.05). In co-culture experiments, NCR-ILC3s frequencies were markedly higher when DCs were derived from CS-exposed mice than from air-exposed mice. This increase was substantially reversed by the addition of EM (P<0.05). Lung NCR-ILC3s frequencies escalate consistently in smokers, COPD patients, and CS-exposed mice. In CS-exposed mice, EM can inhibit DC-mediated NCR-ILC3s activation in the lungs, alleviate CS-related chronic lung inflammation, and ameliorate emphysema.

PMID 42724291
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PubMedJournal of medicinal chemistry2026-09-10

Allosteric Inhibitors of Erythromycin Resistance Methyltransferase Reverse Antibiotic Resistance.

Sahu Damini D, Badgujar Leena Laxmikant LL, Yadav Dhananjay D, Dahm Greta Charlotte GC et al.

Methylation of a critical adenine residue of the 23S rRNA residing in the nascent exit tunnel of the bacterial ribosome, by Erythromycin resistant methyltransferases (Erms), reduces binding of macrolide, lincosamide, and streptogramin B (MLSB) class of antibiotics and confers high-level resistance. Using an allosteric site-directed focused virtual screening approach, nucleoside analogues were identified as the initial scaffold. 6-thioinosine, recognized as a significant initial hit molecule, was confirmed through in vitro screening to be a potent scaffold. Further, structure-based inhibitor evolution approach yielded improved analogues that demonstrated an MIC of 8 μg/mL via a combination therapy approach where Erm inhibitors were administered along with standard antibiotics in MLSB resistant clinical isolates. Our findings demonstrate that a strategy where allosteric inhibitors are developed to impede the ability of pathogenic ribosomal methyltransferases to recognize target RNA can serve as a generic approach for reversal of antibiotic resistance in a combination therapy mode.

PMID 42720463
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PubMedJournal of microbiology & biology education2026-09-09

Modified approach for investigating Prevalence of Antibiotic Resistance in the Environment (PARE)-a research project embedded in lecture-based courses.

Kong Yuwei Y, Hung Wei-Cheng W-C, Jones Adriane A, Bascom-Slack Carol C et al.

The Prevalence of Antibiotic Resistance in the Environment (PARE) Project utilizes standard microbiological methods to engage students in monitoring environmental soil samples for the presence of antibiotic-resistant bacteria. This initiative exemplifies a course-based undergraduate research experience (CURE) within the microbiology curriculum, which has been shown to promote student engagement and persistence in science, technology, engineering, and mathematics (STEM) disciplines by providing opportunities for authentic scientific inquiry. However, broader adoption of PARE can be limited by its requirement for microbiology specialization and biosafety level protocols. To address these barriers, we developed EcPARE (Escherichia coli [E. coli]-specific PARE), a culture-free module of PARE that focuses on detecting pathogenic E. coli in water samples using a modified IDEXX Colilert-18 method. Although IDEXX is primarily designed to detect general fecal contamination, our approach demonstrates its utility as a practical tool for screening erythromycin resistance trends in environmental water samples. In this study, undergraduate participants (n = 47) conducted hypothesis-driven research, including sample collection, laboratory analyses, data analysis, and interpretation. Our findings revealed strong positive correlations between general coliforms or E. coli counts obtained using the modified IDEXX method and total counts from Luria-Bertani plate cultures, indicating concordance between modified IDEXX and conventional plate count methods in the absence of antibiotic selection. This result validates the scientific rigor of our PARE module. Student outcomes assessed through pre- and post-course surveys indicated substantial increases in students' confidence in their scientific skills. Notably, underrepresented students reported greater gains in domains related to sense of community and career confidence, suggesting that such CUREs may be especially impactful for supporting the success and retention of diverse student populations.

PMID 42714158
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PubMedMolecular biology reports2026-09-06

Genomic diversity and resistance determinants of staphylococci from cow and buffalo milk.

Banerjee Jaydeep J, Karim Sk Masud SM, Sharma Deepjyoti D, Choudhury Barnan B et al.

Staphylococci are important mastitis pathogens in dairy animals and serve as reservoirs of antimicrobial resistance genes (ARGs) having zoonotic potential. Genomic characterization of resistant isolates is essential to understand their diversity, resistance mechanisms, and One Health implications. A total of 363 cow and buffalo milk samples-including 108 from animals with mastitis-were screened, yielding 98 staphylococcal isolates, comprising 20 Staphylococcus aureus and 78 coagulase-negative staphylococci (CoNS). Antimicrobial susceptibility testing revealed resistance to cefoxitin (CoNS: 21.7%; S. aureus: 10%), tetracycline (CoNS: 19.2%; S. aureus: 10%), erythromycin (CoNS:16.7%; S. aureus: 10%), gentamicin (CoNS: 10.2%; S. aureus: 10%) and fluoroquinolone (CoNS: 10.2%), while the majority were sensitive to chloramphenicol, cotrimoxazole (~ 95%, each), linezolid (~ 97%), and vancomycin (100%). Nineteen isolates, including two S. aureus, were cefoxitin-resistant, and eight carried the mecA gene. Whole genome sequencing of these eight isolates revealed genome sizes ranging from 2.27 to 2.78 MB, with the methicillin resistant S. aureus (MRSA, ERSST98) isolate possessing the largest genome and the highest rRNA copy number. Comparative genomic analysis revealed various SCCmec types along with an extensive array of resistance determinants, encompassing aminoglycosides, macrolides, tetracyclines, efflux systems, and heavy metals, underscoring the multifaceted resistance repertoire of these strains. Virulence profiling of ERSST98 demonstrated a broad arsenal of adhesins, toxins, and biofilm‑associated genes, highlighting its pathogenic capacity. Mobile genetic elements with diverse plasmid replicons and insertion sequence families further contributed to genomic plasticity. Collectively, this study underscores the genomic diversity of methicillin-resistant staphylococci from dairy animals with extensive resistance determinants and highlights their zoonotic relevance within One Health framework.

PMID 42700195
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PubMedEuro surveillance : bulletin Europeen sur les maladies transmissibles = European communicable disease bulletin2026-09-04

Emerging trends in invasive Streptococcus dysgalactiae subsp. equisimilis infections in Denmark, 2014 to 2024: a nationwide genomic and registry-based study.

Grüttner Jana J, Ronayne Aoife A, Sieber Raphael Niklaus RN, Johannesen Thor Bech TB et al.

BACKGROUNDIncreasing incidence rates of invasive Streptococcus dysgalactiae subspecies equisimilis (iSDSE) have been detected worldwide.AIMWe aimed to investigate iSDSE infection incidence rates in Denmark during 2014-2024, and characterise the genomic population structure of a subset of iSDSE isolates and their antimicrobial resistance (AMR).METHODSUsing national register data, we estimated overall and sex-/age-stratified iSDSE incidences during 2014-2024, by retrospectively identifying cases of invasive infections with group C and G streptococci or S. dysgalactiae (including specified as subspecies equisimilis). From the voluntary national beta-haemolytic streptococci laboratory surveillance system, whole-genome-sequenced isolates from August 2020-September 2022 were used to investigate the iSDSE genomic population structure. Susceptibility to penicillin, erythromycin and clindamycin was determined and AMR genes identified.RESULTSDuring 2014-2024, iSDSE incidence rates increased significantly (linear trend analysis p < 0.001) with mean annual incidence ranging between 10.3 and 16.4 per 100,000, peaking in 2023. Incidence was higher in males, increasing with older age. Nearly 75% of the 1,223 iSDSE isolates belonged to four of 14 genetic clusters. Sequence types (STs) ST20 and ST17 were most prevalent, while emm-type stG62647, a variant associated internationally with higher virulence, dominated. All isolates were phenotypically susceptible to penicillin but approximately 10% were respectively erythromycin and clindamycin resistant. High erythromycin resistance prevalence (57%; 39/68), coinciding with gene ermA, occurred in one genetic cluster.CONCLUSIONThe findings illustrate the need for national registry-based surveillance to detect epidemiological changes and potential outbreaks. Further, continuous genomic surveillance can monitor the occurrence and expansion of genetic clades and AMR genes.

PMID 42695187
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PubMedJournal of dental sciences2026-09-03

Synergistic effects of biodegradable magnesium alloy and erythromycin on osteogenic activity.

Sirisereephap Kridtapat K, Pasanaphong Kitipong K, Osathanon Thanaphum T, Promoppatum Patcharapit P et al.

Biodegradable magnesium (Mg)-based alloys are emerging as promising alternatives to non-resorbable titanium for bone regeneration because of their favorable mechanical properties and biodegradability. However, the interaction between Mg alloys and immunomodulatory agents in promoting osteogenesis remains poorly understood. This study aimed to evaluate the osteogenic effects of an Mg alloy on pre-osteoblasts and to investigate whether erythromycin enhances Mg-induced osteogenic differentiation through regulation of developmental endothelial locus-1 (DEL-1). WE43 Mg alloy disks were immersed in culture medium to produce Mg alloy-conditioned medium at concentrations of 25%, 50%, 75%, and 100%. MC3T3-E1 cells were treated with conditioned medium alone or combined with erythromycin (20 μg/mL). Cell viability was assessed using the MTT assay. Osteogenic differentiation was evaluated by Alizarin Red S staining (ARS), quantitative PCR analysis of osteogenic markers (Runx2, Sp7, Bglap, Edil3), and Western blot analysis of DEL-1 expression. WE43 Mg alloy showed no cytotoxic effects on MC3T3-E1 cells. Treatment with Mg alloy-conditioned medium significantly enhanced osteogenic differentiation and extracellular matrix mineralization. The strongest osteogenic response was observed in cells receiving combined WE43 Mg alloy and erythromycin treatment. DEL-1 expression was significantly upregulated at both mRNA and protein levels in Mg alloy-treated groups, accompanied by increased expression of osteogenic markers. These effects were further amplified by erythromycin supplementation. WE43 Mg alloy promotes osteogenic differentiation of MC3T3-E1 cells, and erythromycin synergistically enhances this effect, potentially via DEL-1 upregulation. These findings support the combined use of immunomodulatory agents and Mg-based biomaterials in regenerative dentistry.

PMID 42688957
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