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pasireotide (Signifor LAR / pasireotide, LAR / pasireotide LAR)

✓ Approved

Novartis AG · SSTR1 · 小分子

什么是 pasireotide?

pasireotide 是一种小分子,由Novartis AG研发。该药已获批,用于治疗相关适应症,给药途径:Injectable (Others)、Intramuscular (IM) Injection、Subcutaneous Injection。

药物档案

商品名Signifor LAR, pasireotide, LAR, pasireotide LAR
公司Novartis AG
药物类别小分子, 多肽类
分子靶点SSTR1, SSTR2, SSTR3, SSTR5
给药途径Injectable (Others), Intramuscular (IM) Injection, Subcutaneous Injection
状态Approved

作用机制

分子靶点

pasireotide 作用于 4 个分子靶点:

SSTR1somatostatin receptor 1 (SS-1-R, SS1-R)
SSTR2somatostatin receptor 2 (SST2)
SSTR3somatostatin receptor 3 (SST3, SS3R)
SSTR5somatostatin receptor 5 (SST5, SS-5-R)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

pasireotide 针对 11 个适应症,涉及 2 个治疗领域。

治疗领域疾病/病症分期
Endocrine disordersAcromegaly✓ Approved
Endocrine disordersPituitary-dependent Cushing's syndrome✓ Approved
Endocrine disordersCarcinoid syndromePhase III
Neoplasms benign, malignant and unspecified (incl cysts and polyps)Colon cancer recurrentPhase III
Neoplasms benign, malignant and unspecified (incl cysts and polyps)Pituitary tumour benignPhase II

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相关研究文献

PubMedJournal of applied clinical medical physics2026-09-10

Comparison of in-field secondary cancer risk based on therapeutic proton dose between proton arc therapy and intensity-modulated proton therapy in lung cancer patients.

Xu Yuankang Y, Chen Wenguang W, Wu Junxiang J, Guo Hao H et al.

Proton arc therapy (PAT) is an emerging delivery modality that delivers proton beams through continuous gantry rotation combined with spot scanning. Compared with intensity-modulated proton therapy (IMPT), PAT improves target conformity and spares organs at risk. However, the dynamic multi-angle irradiation pattern may alter the low-dose region distribution: the low-dose bath expands while the integral dose decreases. The net effect on secondary cancer risk, especially in radiosensitive lungs, remains unclear. Quantitative risk assessment is essential for clinical translation of PAT. To quantitatively compare secondary lung cancer risk between PAT and IMPT using organ equivalent dose (OED) and lifetime attributable risk (LAR) models, and to assess cross-population robustness across China, France, Sweden, and Germany. Data from 25 lung cancer patients (60 Gy/30 fractions) were retrospectively included. For each patient, robustly optimized IMPT and PAT plans were generated with a 3 mm setup and 3% range uncertainties across 21 error scenarios. Dosimetric parameters-ipsilateral lung V 5 , V 20 , and mean dose; whole lungs V 5 , V 20 , and mean dose; and esophageal mean dose-were compared between the two techniques. The mechanistic OED model (with repopulation factor R) and its simplified linear model were used to calculate OED for the ipsilateral lung, both lungs, and the esophagus. LAR was computed by integrating excess absolute risk over the remaining lifetime using patient age, sex, and population-specific parameters (China, France, Sweden, Germany). Relative risk was assessed via the LAR ratio (IMPT/PAT). Paired t-tests or Wilcoxon tests were used with p < 0.05. Under the linear model, PAT produced statistically markedly but modest reductions in absolute LAR for lungs (p < 0.001). Under the mechanistic model, reductions were markedly only in certain populations: ipsilateral lung in France (p = 0.001), Sweden (p < 0.001), Germany (p = 0.003); whole lungs in France (p = 0.046) and Sweden (p = 0.014); but not in China (p = 0.083; p = 1.000) or Germany for whole lungs (p = 0.317). No marked esophageal differences (p > 0.05). LAR ratios were consistent across countries (ipsilateral lung: 1.07-1.09; esophagus: 1.04-1.13), demonstrating robustness. PAT does not increase the modeled in-field secondary cancer risk in the lungs compared with IMPT and shows comparable risk for the esophagus. The risk reduction trend is robust across Chinese and European populations. These findings suggest that PAT does not increase modeled secondary lung cancer risk compared with IMPT and may even provide a modest risk reduction, providing quantitative evidence for clinical application.

PMID 42717736
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PubMedVox sanguinis2026-09-09

Association of acute normovolemic hemodilution with hematologic inflammatory indices and early clinical outcomes after coronary artery bypass grafting.

Yamac Dilek Metin DM, Yilmaz Yadigar Y, Erturk Tuna T, Emirkadi Hakan H et al.

Acute normovolemic hemodilution (ANH) is an established patient blood management strategy in cardiac surgery, but its effects on postoperative inflammatory biomarkers remain unclear. In this study, we evaluate the association of ANH with inflammatory indices, lactate-to-albumin ratio, transfusion requirements, and early postoperative outcomes after coronary artery bypass grafting (CABG). This retrospective, single-center study included 366 patients who underwent elective isolated CABG with cardiopulmonary bypass. Patients were assigned to an ANH group (n = 169) or a control group (n = 197). Primary outcomes were postoperative neutrophil-to-lymphocyte ratio (NLR), platelet-to-lymphocyte ratio (PLR), neutrophil-to-monocyte-to-lymphocyte ratio (NMLR), and lactate-to-albumin ratio (LAR). Secondary outcomes included blood transfusion, intraoperative bleeding, mechanical ventilation, intensive care unit (ICU) stay and hospital stay, postoperative complications, and infections. No significant differences were observed in NLR, PLR, or NMLR between the groups. LAR was significantly lower in the ANH group (0.31 ± 0.12 vs. 0.51 ± 0.93, p < 0.001). ANH was also associated with lower blood product utilization, reduced intraoperative bleeding, shorter duration of mechanical ventilation, shorter ICU stay and hospital stay, and lower rates of postoperative complications and infections (all p < 0.05). In patients undergoing CABG, ANH was associated with improved early postoperative outcomes and a lower LAR but not with significant changes in routine hematologic inflammatory indices. These findings suggest that the benefits of ANH may extend beyond blood conservation.

PMID 42716536
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PubMedJournal of the American Medical Directors Association2026-09-09

Routine Hematologic Indices as Scalable Biomarkers for Frailty: A Comprehensive Systematic Review and Meta-Analysis.

Yang Yan-Wu YW, Gao Li L, Zhang Yan Y, Wan Zhi Z et al.

To systematically evaluate the associations of albumin-based biomarkers, including the C-reactive protein-to-albumin ratio (CAR/hsCAR), neutrophil percentage-to-albumin ratio (NPAR), lactate-to-albumin ratio (LAR), and C-reactive protein-albumin-lymphocyte (CALLY) index, with mortality and major adverse cardiovascular events (MACE) in patients with coronary artery disease (CAD), and to compare their prognostic and discriminative performance. Systematic review and meta-analysis. Thirty-four studies involving 47,763 patients with CAD were included, encompassing predominantly acute coronary syndrome (ACS)-related populations as well as broader coronary and cardiovascular cohorts. We systematically evaluated albumin-based biomarkers, including CAR/hsCAR, NPAR, LAR, and CALLY. Pooled associations with mortality and MACE were estimated using effect measures reported by the original studies. Discriminative performance and potential clinical utility were also evaluated where data were available. Higher CALLY values were associated with lower all-cause mortality (HR 0.46, 95% CI 0.24-0.87) and showed a directionally protective but nonsignificant association with MACE (HR 0.44, 95% CI 0.18-1.08). Elevated CAR/hsCAR was associated with increased mortality (OR 1.61, 95% CI 1.09-2.38) and MACE (HR 1.37, 95% CI 1.21-1.56) in ACS-related cohorts. NPAR showed the most consistent association with mortality (HR 1.88, 95% CI 1.71-2.08; I² = 4.8%), whereas its association with MACE was less stable (HR 1.86, 95% CI 0.56-6.13). LAR showed the largest pooled effect estimate for mortality (HR 2.50, 95% CI 1.78-3.51). In discriminative analyses, CAR showed the most balanced performance for long-term MACE, NPAR showed the strongest rule-in profile for long-term MACE, and CAR and CALLY showed the best discrimination for mortality. Albumin-based biomarkers are associated with adverse outcomes in CAD, particularly in ACS-related populations, with distinct prognostic patterns across biomarkers and clinical endpoints. These routinely available indices may provide complementary information for risk stratification; however, prospective studies are needed to determine their incremental prognostic value and clinical utility beyond established risk assessment approaches.

PMID 42715816
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PubMedFrontiers in medicine2026-09-08

Lactate-to-albumin ratio improves prediction of perioperative mortality in lung transplant patients.

Yi Yu Y, Luo Ge G, Wang Ying Y, Ran Xinhong X et al.

Perioperative mortality remains elevated among lung transplant recipients. The lactate-to-albumin ratio (LAR) is a prognostic indicator, but its role in predicting mortality in lung transplant patients remains unclear. The study aims to assess the incremental prognostic value of LAR and develop a more accurate prediction model for perioperative mortality in lung transplant patients. This study conducted a single-center, retrospective analysis involving 379 lung transplant recipients. A base model was developed to predict 30-day postoperative mortality and a modified model was then constructed by incorporating LAR. Model performance was evaluated using the area under the curve (AUC), Brier score, and calibration curves. DeLong and likelihood ratio tests compared models, while continuous Net Reclassification Improvement (NRI) and Integrated Discrimination Improvement (IDI) quantified accuracy improvements. Of 379 patients, 51 (13.46%) died within 30 days post-transplant. LAR was found to be an independent predictor of perioperative mortality in lung transplant patients. Other predictors in the modified model included blood transfusion, cold ischemia time, and fluid balance. The inclusion of LAR significantly improved the modified model's discriminatory ability (AUC: 0.807 vs. 0.764; p = 0.024) and calibration (Brier score: 0.0927 vs. 0.1025). The likelihood ratio test confirmed a significantly improved model fit (p < 0.0001). The continuous NRI and IDI were 0.643 and 0.090, respectively (p < 0.001). A nomogram and an interactive web-based tool were developed to facilitate individualized risk assessment. The modified model incorporating LAR provides a more accurate and comprehensive assessment of perioperative mortality risk.

PMID 42707950
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PubMedRadiation protection dosimetry2026-09-08

Lifetime attributable cancer risk assessment in pediatric patients undergoing I-124 PET for differentiated thyroid cancer.

Maddahi Amirhossein A, Hosseinabadi Roghiye Bodaghi RB, Talebi Asra Sadat AS

The increasing use of I-124 PET for differentiated thyroid cancer (DTC) has raised concerns about radiation exposure in pediatric patients because of their radiosensitivity. This study estimated organ-absorbed doses and the lifetime attributable risk (LAR) of secondary cancer following I-124 PET using Monte Carlo simulations with pediatric voxel phantoms representing 10- and 15-year-old males and females. Organ doses were calculated for oral and intravenous administration under different thyroid uptake conditions, and LAR was estimated using the Biological Effects of Ionizing Radiation (BEIR) VII model. The thyroid absorbed dose was slightly higher after intravenous administration, whereas the total-body dose depended mainly on age. Younger patients showed nearly twice the LAR of older patients. Females had a higher solid cancer risk, whereas leukemia risk was greater in males. Thyroid uptake and administration route had minimal effect on LAR. These findings support individualized I-124 PET protocols to maximize diagnostic benefit while minimizing long-term radiation risk in pediatric DTC.

PMID 42709686
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PubMedThe Eurasian journal of medicine2026-09-07

Association of Early and Late Postnatal Serum Lactate/Albumin Ratio and Retinopathy of Prematurity in Preterm Infants: A 2 Time Point Comparative Study.

Çalışkan Büşra B, Korkut Dilara D, Kara Mustafa M, Tekgündüz Kadir Şerafettin KŞ

One easily accessible compound index that shows the metabolic and inflammatory status of critically ill patients is the lactate-albumin ratio (LAR). This study set out to evaluate the connection between LAR and retinopathy of prematurity (ROP) in premature infants. The investigation was conducted retrospectively on 150 premature infants born before 34 weeks who underwent screening for ROP in the neonatal intensive care unit. Demographic and clinical data, as well as ROP examination findings, were recorded for all participants. For the first 24 h following delivery (early phase) and at 34-36 weeks' postmenstrual age (late period), serum lactate and albumin values were measured separately. For each of these measurements, the lactate/albumin ratio was calculated. Mann-Whitney U-test, logistic regression, correlation analyses, together with receiver operating characteristic (ROC) analysis were performed. In infants who developed ROP, both the LAR calculated in the early phase (1.16 ± 0.56, P = .03) and the LAR calculated in the late period (0.53 ± 0.19, P = .02) were found to be significantly higher than those without ROP. In post hoc analyses based on disease severity, LAR values were significantly higher in the treatment-requiring ROP group (P = .02). In logistic regression, late-period LAR showed a borderline but statistically non-significant association with ROP development (OR = 11.05; 95% CI = 0.97-125.9; P = .053). Lactate-albumin ratio values were associated with ROP development and disease severity in premature infants. However, LAR was not demonstrated to be an independent predictor of ROP in the present study. As a composite index reflecting nutrition, inflammation, tissue oxygenation, and metabolic stress, LAR may provide complementary information regarding systemic vulnerability in premature infants rather than serving as a standalone predictive or screening biomarker. Further prospective and multicenter studies are needed to clarify its potential role in ROP risk assessment. Cite this article as: Çalışkan B, Korkut D, Kara M, Tekgündüz KŞ. Association of early and late postnatal serum lactate/albumin ratio and retinopathy of prematurity in preterm infants: a 2 time point comparative study. Eurasian J Med. 2026, 58(4), 1457, doi: 10.5152/eurasianjmed.2026.261457.

PMID 42703816
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