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rituximab (Kikuzubam / PBO326)

✓ Approved

Probiomed · MS4A1 · 单克隆抗体

什么是 rituximab?

rituximab 是一种单克隆抗体,由Probiomed研发。该药已获批,用于治疗相关适应症,给药途径:Injectable (Others)、Intracerebral/cerebroventricular Injection、Intravenous (IV)、Subcutaneous Injection。

药物档案

商品名Kikuzubam, PBO326
公司Probiomed
药物类别单克隆抗体, 抗体
分子靶点MS4A1
给药途径Injectable (Others), Intracerebral/cerebroventricular Injection, Intravenous (IV), Subcutaneous Injection
状态Approved

作用机制

分子靶点

rituximab 作用于 1 个分子靶点:

MS4A1membrane spanning 4-domains A1 (S7, B1)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

rituximab 针对 8 个适应症,涉及 4 个治疗领域。

治疗领域疾病/病症分期
Neoplasms benign, malignant and unspecified (incl cysts and polyps)B-cell lymphoma✓ Approved
Neoplasms benign, malignant and unspecified (incl cysts and polyps)Chronic lymphocytic leukaemia✓ Approved
Neoplasms benign, malignant and unspecified (incl cysts and polyps)Diffuse large B-cell lymphoma✓ Approved
Neoplasms benign, malignant and unspecified (incl cysts and polyps)Non-Hodgkin's lymphoma✓ Approved
Musculoskeletal and connective tissue disordersRheumatoid arthritis✓ Approved

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相关研究文献

PubMedCureus2026-07-27

De Novo Proliferative Glomerulonephritis With Monoclonal Immunoglobulin Deposits (PGNMID) in a Renal Transplant Recipient.

Murugesan Ram Prabahar RP, Sivanandam Sathiyan S, Jayam Jayanivash J, Kurian Anila A AA

Proliferative glomerulonephritis with monoclonal immunoglobulin deposits (PGNMID) represents a distinct glomerular pathology, classified under monoclonal gammopathy of renal significance (MGRS). In renal transplant, PGNMID usually develops as a recurrent disease, but can rarely arise de novo. Recurrence is relatively common, typically appearing within five to six months post-transplant, and is linked to poor graft outcomes. De novo PGNMID is exceedingly rare, with few reported in the literature. It generally presents in the late post-transplant period, with a more indolent clinical course and a variable response to immunotherapy. This case report is of a 50-year-old patient who had diabetic nephropathy as his native kidney disease. This report documents a unique instance of de novo PGNMID, occurring three years post-transplantation with persistent allograft dysfunction. The transplant kidney biopsy showed mesangial hypercellularity with immunoglobulin (Ig)G and kappa light chain deposition by immunofluorescence; however, electron microscopy was non-contributory due to the absence of viable glomeruli. Despite extensive evaluation, we could not identify any clone contributing to the MGRS in the bone marrow, nor could we identify any other evidence of lymphoproliferative disease on positron emission tomography-computed tomography (PET-CT). We managed the patient with empirical clone-directed therapy against a likely B-cell clone using Rituximab. During rituximab therapy, the patient developed E. coli urosepsis, which was managed successfully. At the last follow-up, graft function remained stable without progression, although the duration of follow-up is limited.

PMID 42504369
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PubMedCurrent oncology (Toronto, Ont.)2026-07-27

Prognostic Value of Semi-Quantitative Metabolic Parameters on [18F]FDG PET/CT in Patients with Diffuse Large B-Cell Lymphoma at Diagnosis.

Cencini Emanuele E, Orsini Federica F, Franceschini Marta M, Fredducci Sara S et al.

After first-line therapy with rituximab, cyclophosphamide, doxorubicin, vincristine, and prednisone (R-CHOP), 20-30% of patients with diffuse large B-cell lymphoma (DLBCL) have relapsed or refractory disease. Semi-quantitative volume parameters on [18F]Fluorodeoxyglucose positron emission tomography/computed tomography ([18F]FDG PET/CT), performed at diagnosis, could represent variables with prognostic influence. We retrospectively analyzed 53 consecutive patients, treated between 2016 and 2022. Semi-quantitative metabolic parameters, assessed by the software LIFEx, included total metabolic tumor volume (TMTV), total lesion glycolysis (TLG), Dmax and DmaxVox. All cases received R-CHOP/CHOP-like regimens with curative intent. The International Metabolic Prognostic Index (IMPI) was low in 43/53 cases (81.1%). CR was achieved in 49/53 patients (92.4%); 7/53 (13.2%) relapsed after achieving a CR. For the entire cohort, 2-year PFS and OS were 84.9% and 90.6%, respectively, while 5-year PFS and OS were 65.5% and 77.6%, respectively. IPI score, B symptoms, TMTV, Dmax and DmaxVox were associated with reduced PFS in an exploratory univariate analysis. IPI score was the only variable for which we found a significant association with reduced OS. In this exploratory analysis in a small, event-limited population, we suggest the baseline, semi-quantitative metabolic parameters of PET/CT at diagnosis could contribute to defining tumor burden and to predict PFS for DLBCL patients.

PMID 42505194
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PubMedClinica chimica acta; international journal of clinical chemistry2026-07-27

Diagnostic pitfall: NSAID-induced membranous nephropathy with PLA2R positivity, IgG1-predominant deposits, C1q positivity, and concurrent acute interstitial nephritis-A case report.

Li Jingzhen J, Zhang Qianqian Q, Chen Zhengyue Z, Qiu Yingyin Y et al.

Serum anti-phospholipase A2 receptor (PLA2R) antibody is widely used to diagnose primary membranous nephropathy (MN), but PLA2R positivity also occurs in secondary MN, especially nonsteroidal anti-inflammatory drug (NSAID)-induced MN, leading to a common diagnostic pitfall. We report a 71-year-old female with long-term unsupervised NSAID administration for polymyalgia rheumatica, presenting with recurrent nephrotic syndrome and acute kidney injury. Initial laboratory tests revealed severe hypoalbuminemia (15.7 g/L), elevated serum creatinine (3.98 mg/dL), massive proteinuria (10.24 g/24 h), and positive anti-PLA2R antibody (39.69 U/mL). The etiology of her first nephrotic episode remained unclear, and renal biopsy during disease relapse finally confirmed NSAID-induced secondary MN. Pathological examination demonstrated PLA2R-positive MN with immunoglobulin G1 (IgG1)-predominant immune deposits, moderate (2+) glomerular complement component 1q (C1q) deposition, and concomitant severe acute interstitial nephritis. The patient achieved clinical remission after NSAID discontinuation and treatment with intravenous methylprednisolone combined with rituximab, but disease relapse occurred after inadvertent NSAID re-exposure. This case highlights that PLA2R positivity does not exclude drug-induced secondary MN. IgG subclass profiling and C1q staining are critical complementary biomarkers for precise differential diagnosis and can effectively prevent the common diagnostic pitfall of attributing PLA2R positivity exclusively to primary MN. Permanent NSAID discontinuation remains the cornerstone of disease management.

PMID 42503368
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PubMedMedical sciences (Basel, Switzerland)2026-07-27

Primary Lymphomas of the Female Genital Tract: Recognizing the Rare Mimicker of Gynecologic Malignancy.

Stavros Sofoklis S, Daskalaki Maria-Anastasia MA, Dafopoulos Stefanos S, Moustakli Efthalia E et al.

Primary lymphomas of the female genital tract (PLFGT) are extremely rare neoplasms, representing a minor fraction of both extranodal lymphomas and gynecologic malignancies. Due to their nonspecific clinical presentation and overlapping imaging features with more common gynecologic tumors, diagnosis is often delayed or missed. This narrative review aims to synthesize current evidence on the clinical characteristics, histologic subtypes, diagnostic approaches, treatment strategies, and prognostic factors of PLFGT, emphasizing recent developments that may influence clinical practice. A comprehensive literature review was conducted, incorporating data from institutional case series, population-based studies, and recent genomic investigations focusing on PLFGT across various anatomical sites: ovary, uterus, cervix, and vagina. PLFGT typically affects women aged 44-68 years, with the ovary being the most frequently involved organ. The most common subtype is diffuse large B-cell lymphoma (DLBCL), followed by Burkitt lymphoma and marginal zone lymphoma. Patients usually present with pelvic pain, mass, or abnormal bleeding, while B symptoms are infrequent. Image-guided core needle biopsy has emerged as a valuable diagnostic approach that may reduce unnecessary surgery. Characteristic sonographic findings, such as hypoechoic, well-defined lesions and homogeneous uterine echo reduction, should raise clinical suspicion, though primary and metastatic disease cannot be distinguished solely by imaging. Rituximab-containing regimens (R-CHOP) are the mainstay of treatment and have improved outcomes. Despite treatment, central nervous system (CNS) recurrence remains a concern, particularly in ovarian involvement. Additionally, mutations in MYD88 and CD79B, although not prognostic, offer potential for personalized therapy. Timely diagnosis and appropriate systemic therapy are critical for improving survival in PLFGT. Advances in imaging, biopsy techniques, and molecular profiling are reshaping the diagnostic and therapeutic landscape of this rare but clinically significant disease.

PMID 42506377
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PubMedMultiple sclerosis journal - experimental, translational and clinical2026-07-26

Family planning and multiple sclerosis - part 2: Does real-world practice align with Swedish treatment guidelines?

Machado Alejandra A, Pettersson Emma E, Teni Fitsum Sebsibe FS, Friberg Emilie E et al.

Managing family planning and treatment in women with multiple sclerosis (MS) requires balancing disease control with medication safety. Despite guidelines, practice often adapts to individual needs, with clinicians adjusting disease-modifying therapies (DMTs) to protect maternal and fetal health. This study examines pregnancy-related MS treatment in Sweden. We identified 130 women (153 pregnancies) from a 2021 online MS questionnaire and linked responses to the Swedish MS register to capture DMT use during three periods: 25 weeks before conception, pregnancy (≈40 weeks), and 25 weeks postpartum. DMTs were classified as "accepted," "discontinuation recommended"-requiring monitoring, or "not recommended" in planned pregnancy. Before conception, among 153 pregnancies, 26% involved DMTs considered acceptable before and during pregnancy, while 55% involved DMTs for which discontinuation before conception is recommended-of which rituximab accounted for nearly half of all pregnancies (47%, n = 72). Three percent were exposed to ´not recommended´ DMTs, and 16% had no prior treatment. Overall, 29% discontinued DMTs before or shortly after conception, while 58% (n = 88) had ongoing or recent treatment exposure, defined as treatment administered within 6 months before conception or, in a minority of cases, after conception. Among these, 50% (n = 77) involved rituximab-and 13% remained untreated. Postpartum, 58% resumed treatment, 3% remained under long-lasting DMT effects, and 39% did not initiate DMT, likely due to breastfeeding. Overall, real-world practice in Sweden broadly aligns with national recommendations, with widespread use of rituximab before pregnancy reflecting its perceived safety and durable effect, alongside some individualized deviations from discontinuation guidance.

PMID 42502707
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PubMedJHEP reports : innovation in hepatology2026-07-26

Post-transplant alloimmune liver disease in bile salt export pump deficiency: A multicenter study.

Gardin Antoine A, Rubino Chiara C, Michaut Alice A, Résin Géraldine G et al.

Patients with severe bile salt export pump (BSEP) deficiency may develop alloimmune anti-BSEP liver disease (AIBD) after liver transplantation (LT) due to anti-BSEP antibodies, but its frequency and risk factors are not precisely known. A multicentre cohort of 35 patients who underwent LT for severe BSEP deficiency was screened retrospectively or prospectively after 2010 for anti-BSEP antibodies. Risk factors, management and outcome of AIBD were analysed. Ten patients (29%) were screened positive for anti-BSEP antibodies and all developed AIBD, in median 5 years (range: 1.5-14) after LT. Clinical remission of AIBD was achieved in nine patients using various immunosuppressive therapies, with decreased or negative anti-BSEP antibody titers in six patients, all having received rituximab or plasmapheresis/immunoadsorption. Relapse occurred in six patients out of nine, although maintenance therapy using rituximab and/or immunoglobulins enabled prolonged relapse-free survival. Because of AIBD, six patients (60%) required liver retransplantation either at initial AIBD episode or at relapse, and three patients (30%) died. Among the 25 patients without AIBD, one died (4%) and another one was retransplanted (4%). While a severe ABCB11 genotype (biallelic truncating variants) was significantly associated with AIBD (80% in patients with AIBD vs 28% in patients without AIBD, p=0.008), negative BSEP immunostaining on native liver, post-LT CMV infection, presence of biliary anastomosis strictures or graft rejection were not. In patients with severe BSEP deficiency, AIBD is a frequent post-LT complication that should be screened for, especially in patients with severe ABCB11 genotypes. Early diagnosis and the use of rituximab and plasmapheresis/immunoadsorption may improve patient outcome. Alloimmune anti-BSEP liver disease is a frequent and severe complication after liver transplantation in patients with BSEP (Bile Salt Export Pump) deficiency, affecting nearly one-third of recipients in this multicentre cohort study. Patients carrying biallelic protein-truncating ABCB11 variants are at particularly high risk and should undergo systematic post-transplant screening for anti-BSEP antibodies. Early recognition of alloimmune anti-BSEP liver disease and timely treatment with B-cell-depleting and antibody-removal therapies, including rituximab and plasmapheresis/ immunoadsorption, may improve outcomes and reduce graft loss. These findings support the implementation of structured surveillance strategies and risk-adapted management in this rare but life-threatening condition.

PMID 42501969
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