Drug Database
GR

granulocyte colony stimulating factor (Hebervital)

✓ Approved

Heber Biotec · CSF3 · 重组蛋白

什么是 granulocyte colony stimulating factor?

granulocyte colony stimulating factor 是一种重组蛋白,由Heber Biotec研发。该药已获批,用于治疗相关适应症,给药途径:Injectable (Others)。

药物档案

商品名Hebervital
公司Heber Biotec
药物类别重组蛋白
分子靶点CSF3
给药途径Injectable (Others)
状态Approved

作用机制

分子靶点

granulocyte colony stimulating factor 作用于 1 个分子靶点:

CSF3colony stimulating factor 3 (GCSF, CSF3OS)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

granulocyte colony stimulating factor 针对 2 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Blood and lymphatic system disordersNeutropenia✓ Approved
Blood and lymphatic system disordersBone marrow disorder✓ Approved

相关研究文献

PubMedBritish journal of haematology2026-09-10

A pro-inflammatory cytokine signature characterises thrombotic antiphospholipid syndrome despite stable anticoagulation.

Ducker Catherine B CB, Preece Megan V MV, Schofield Jeremy J, Pericleous Charis C et al.

Inflammation contributes to primary antiphospholipid syndrome (PAPS) pathogenesis, but cytokine profiles and associated thrombotic phenotypes remain incompletely defined. A panel of 20 cytokines, chemokines and endothelial activation markers was analysed in 37 PAPS patients on stable anticoagulation and 12 healthy controls (HC). We compared concentrations between groups and performed unsupervised hierarchical clustering and principal component analysis (PCA) to identify inflammatory subgroups. Compared with HC, patients with PAPS exhibited significantly elevated levels of 14/20 analytes: granulocyte-macrophage colony-stimulating factor (GM-CSF), interferon (IFN)-γ, interleukin (IL)-1α, IL-1β, IL-6, IL-10, IL-12p70, IL-13, IL-17a, tumour necrosis factor-α (TNF-α), intercellular adhesion molecule-1 (ICAM-1), P-selectin and macrophage inflammatory protein-1β (MIP1β) (all p < 0.05). Unsupervised clustering identified three inflammatory antiphospholipid syndrome (APS) subgroups distinct from HC. A core cytokine signature comprising GM-CSF, IL-6, IL-10, IL-12p70, IL-13 and TNF-α was elevated across all APS clusters. One cluster, enriched for arterial thrombosis, demonstrated a more pronounced inflammatory phenotype, with increased IFN-α. Comparison of phenotypes showed significantly higher concentrations of GM-CSF, IFN-α, IL-1α, IL-4, IL-6, IL-10, IL-17a and TNF-α in arterial versus venous thrombosis. Our findings demonstrate widespread cytokine dysregulation and distinct inflammatory subgroups in PAPS, with arterial thrombosis showing stronger inflammation than venous thrombosis, supporting divergent thrombo-inflammatory mechanisms and potential precision immunomodulatory therapeutic targets.

PMID 42717283
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PubMedFrontiers in oncology2026-09-10

Umbilical cord blood infusion enhances hematopoietic recovery and improves survival in elderly AML patients with chemotherapy-induced myelosuppression: a retrospective study.

Zhou Yimin Y, Ren Yuye Y, Zhang Lan L, Hu Wenya W et al.

Elderly AML (Acute Myeloid Leukemia) patients exhibit increased mortality owing to chemotherapy-induced myelosuppression. Umbilical cord blood (UCB) contains hematopoietic stem/progenitor cells and a spectrum of regenerative cytokines that actively promote hematopoietic regeneration. We investigated whether umbilical cord blood (UCB) infusion enhances hematopoietic recovery in elderly AML patients who experience chemotherapy-induced myelosuppression during post-chemotherapy supportive care. We retrospectively analyzed 95 elderly patients with AML in complete remission (CR1) who previously developed grade III-IV chemotherapy-induced myelosuppression. The control group (n=60) received standard supportive care, including granulocyte colony-stimulating factor (G-CSF), blood product transfusions, and antibiotic therapy. The experimental group (n = 35) underwent infusion of unrelated umbilical cord blood (UCB; CD34+ cells ≥2×106/kg) within 24 hours post - chemotherapy, along with standard supportive care. Neutrophil recovery duration (≥1.0×109/L) was reduced in the UCB group (16 VS 23 days, P<0.01). Platelet recovery (≥50×109/L) was also shorter (13 days vs. 19 days, P<0.01), though hemoglobin recovery (≥70 g/L) did not differ significantly (18 days vs. 21 days, P>0.05). The incidence of grade III-IV infections decreased to 31.43% (vs. 55.00%, P<0.05), that of bleeding events decreased to 11.43% (vs. 33.33%, P<0.05), that of transfusion-related allergic reactions decreased to 17.14% (vs. 26.67%, P<0.05), and chemotherapy delay/reduction rates decreased to 14.29% (vs. 35.00%, P<0.05). The overall survival (OS) was significantly longer in the UCB group, and the 2-year relapse-free survival (RFS) was higher (P<0.05). The most common adverse events were transfusion-related (e.g., rash and transient fever). Graft-versus-host disease (GVHD) was not observed in the UCB group.These findings indicate that UCB infusion enhances hematopoietic recovery, reduces complications, and improves the survival of elderly patients with AML after chemotherapy, likely through the synergistic effects of CD34+ cells and cytokines.

PMID 42718531
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PubMedAnnals of translational medicine2026-09-10

Tumor microenvironment and signaling pathways in melanoma brain metastasis.

Rosell Rafael R, González-Cao María M, Olmo-González Daniel D, Hold Emilia E et al.

Melanoma has one of the highest propensities to metastasize to the brain, and despite major advances with immune checkpoint inhibitors, brain metastases remain a leading cause of morbidity and mortality. The biological mechanisms governing brain colonization, immune evasion, and resistance to therapy are incompletely understood. This review summarizes recent advances in the understanding of the tumor microenvironment and signaling pathways involved in melanoma brain metastasis, with emphasis on mechanisms that may provide novel therapeutic opportunities. We performed a review of preclinical and clinical studies investigating molecular pathways, immune-cell interactions, and metabolic programs associated with melanoma brain metastasis and response to immunotherapy. Emerging evidence identifies enhancer of zeste homolog 2 (EZH2) phosphorylation by Src kinase as a key driver of brain metastasis through granulocyte colony-stimulating factor (G-CSF) production and recruitment of immunosuppressive neutrophils. Microglia and tumor-associated macrophages constitute major components of the brain metastatic microenvironment and actively support tumor progression. Spleen tyrosine kinase (Syk) signaling contributes to microglial activation and immune-related neurotoxicity during anti-programmed death 1 (PD-1) therapy. Mitochondrial dysfunction, including alterations in mitochondrial contact site and cristae organizing system (MICOS) complex components such as Mic19 and Mic60, promotes innate immune signaling through cyclic GMP-AMP synthase (cGAS)-stimulator of interferon genes (STING) and TANK-binding kinase 1 (TBK1). TBK1 emerges as a central regulator linking neuroinflammation, microglial activation, metastatic progression, and therapeutic resistance. In addition, metabolic reprogramming mediated by tectonic family member 1 (TCTN1) and carnitine palmitoyltransferase 1A (CPT1A) enhances fatty acid oxidation and promotes melanoma metastasis. These pathways may represent actionable targets that complement immune checkpoint blockade. Melanoma brain metastasis is driven by complex interactions between tumor cells, neutrophils, microglia, and mitochondrial signaling networks. Src-EZH2, TBK1-dependent inflammatory pathways, and TCTN1/CPT1A-mediated metabolic reprogramming are emerging biomarkers and therapeutic targets. Integrating these approaches with anti-PD-1 and anti-cytotoxic T-lymphocyte-associated protein 4 (CTLA-4) therapies may improve disease control, overcome resistance, and reduce immune-related adverse events in patients with melanoma brain metastases.

PMID 42719252
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PubMedBritish journal of haematology2026-09-10

Optimizing cord blood unit selection to improve survival after single-unit unrelated cord blood transplantation for adult myelodysplastic syndrome.

Konuma Takaaki T, Fujioka Machiko M, Fuse Kyoko K, Suwabe Tatsuya T et al.

Unrelated cord blood transplantation (CBT) is an important alternative donor option for adult patients with myelodysplastic syndrome (MDS); however, the prognostic significance of cord blood unit characteristics following CBT remains unclear and may vary according to disease risk. We conducted a nationwide retrospective study of 1767 adult patients with MDS who underwent first single-unit CBT between 1999 and 2023, including 529 patients with low-risk and 1238 with high-risk disease at transplantation. Cord blood unit characteristics were not significantly associated with disease-free survival (DFS) in patients with low-risk MDS. In contrast, in patients with high-risk MDS, higher cryopreserved cluster of differentiation (CD)34+ cell dose and higher colony-forming unit-granulocyte/macrophage dose were associated with improved DFS, whereas human leucocyte antigen (HLA) serological one-locus mismatch and female-to-male donor-recipient sex mismatch were independently associated with inferior DFS. Restricted cubic spline Cox regression demonstrated a significant non-linear association between CD34+ cell dose and DFS, as well as relapse, in high-risk MDS. These findings demonstrate that the prognostic impact of cord blood unit characteristics after single-unit CBT differs according to MDS risk status and support a risk-adapted approach to cord blood unit selection, particularly for patients with high-risk MDS.

PMID 42717739
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PubMedGeneral physiology and biophysics2026-09-10

Transcription factor KLF4 suppresses the malignant progression of colorectal cancer by activating ETFDH transcription.

Zeng Yan Y, Liu Qiaozhen Q, Xu Yali Y, Zhao Tong T et al.

Colorectal cancer (CRC) is a common cause of cancer-related deaths worldwide. Electron transfer flavoprotein dehydrogenase (ETFDH) is a novel prognostic biomarker for human CRC. However, the role and molecular mechanism of ETFDH in CRC are still unclear. DEGs in CRC development were identified using mRNA microarray datasets GSE23011, GSE44076, and GSE113513. Gene expression was determined using RT-qPCR and Western blot. Cell proliferation, migration, and invasion were detected by EdU, Colony formation, Transwell, and wound healing. Effects of CRC cells on CD8+ T cell apoptosis were analyzed using flow cytometry. Effects of ETFDH on CRC cell growth in vivo was analyzed using xenograft model. After JASPAR prediction, the binding between Transcription factor Kruppel-like factor 4 (KLF4) and ETFDH promoter was verified using ChIP and dual-luciferase reporter. ETFDH and KLF4 were decreased in CRC tissues and cells. ETFDH upregulation blocked CRC cell proliferation, migration, invasion, and repress the apoptosis of CD8+ T cells in vitro. ETFDH overexpression hindered CRC tumor growth in vivo. Mechanistically, KLF4 enhanced the transcriptional activity of ETFDH via binding to its promoter region. KLF4-activated ETFDH transcription suppresses CRC cell malignant behavior and decreases the apoptosis of CD8+T cells, which provides a promising therapeutic target for CRC.

PMID 42717785
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PubMedAnnals of translational medicine2026-09-10

Screening for atrial fibrillation according to serum thyroid-stimulating hormone: an opportunity for refinement?

Mavilakandy Akash Kamalakshan AK, Lip Gregory Y H GYH

PMID 42719254
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