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prasterone (Mylis)

✓ Approved

Merck & Co. · AR · 小分子

什么是 prasterone?

prasterone 是一种小分子,由Merck & Co.研发。该药已获批,用于治疗相关适应症。

药物档案

商品名Mylis
公司Merck & Co.
药物类别小分子
分子靶点AR
状态Approved

作用机制

分子靶点

prasterone 作用于 1 个分子靶点:

ARandrogen receptor (DHTR, AR8)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

prasterone 针对 1 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Surgical and medical proceduresLabour induction✓ Approved

相关研究文献

PubMedCells2026-07-27

Exploratory Metabolomic Profiling of Plasma and Cerebrospinal Fluid in a Pilot Study of Children with Acute Lymphoblastic Leukemia.

Wasilewski Andrzej A, Czapor-Irzabek Hanna H, Ściskalska Milena M, El Idrissi Adam A et al.

Acute lymphoblastic leukemia (ALL) is the most common pediatric malignancy and is associated with profound metabolic reprogramming. This exploratory study aimed to characterize the metabolomic profiles of plasma and cerebrospinal fluid (CSF) in children with newly diagnosed pre-B-cell acute lymphoblastic leukemia (pre-B ALL) prior to therapy. Metabolomic analyses were performed using mass spectrometry-based platforms combined with multivariate statistical approaches (PCA, OPLS-DA, SVM-RFE, EBAM). In plasma, we identified 41 significantly altered metabolites (FDR < 0.011), revealing a distinct signature that differentiated pre-B ALL patients from healthy controls. Specifically, patients exhibited elevated levels of hypoxanthine, xanthine, and phosphatidylcholine derivatives, alongside reduced concentrations of L-cysteine and prasterone sulfate, indicating systemic dysregulation of purine, lipid, and amino acid metabolism. In CSF, we observed a distinct metabolic profile characterized by coordinated disturbances in purine degradation, phospholipid metabolism, and sphingolipid pathways. Notably, correlation analysis between the two matrices suggested that systemic metabolic shifts, particularly in purine metabolism (e.g., hypoxanthine and xanthine levels), are mirrored within the central nervous system microenvironment. These findings indicate that children with pre-B ALL exhibit specific metabolic alterations in both compartments before treatment. This work serves as a proof-of-concept for applying metabolomics in pediatric oncology, highlighting the necessity for further validation in larger, prospective cohorts to assess the clinical utility of these profiles.

PMID 42505365
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PubMedEcological applications : a publication of the Ecological Society of America2026-07-26

Free-ranging livestock grazing shifts the acoustic community in a northeast Asian temperate forest.

Wang Shizheng S, Wei Xintong X, Jia Kangning K, Ma Xiao X et al.

Understanding livestock-wildlife interactions, especially in forest ecosystems, is critical for biodiversity conservation and sustainable land management. However, the long-term and cascading impacts of livestock grazing on forest structure and community bioacoustics are important yet largely neglected areas of research. Here, we used acoustic indices and a sound event detection (SED) model to evaluate the effects of continuous cattle grazing on seasonal soundscapes in Northeast China. We collected and analyzed over 18,785 h of recordings from 10 cattle-grazed forest plots and 10 ungrazed forest plots in Northeast China. We identified sound events in each recording via deep learning and calculated six acoustic indices, as well as extracted vegetation characteristics using light detection and ranging point cloud data. Our results revealed that grazing activities significantly changed seasonal soundscape dynamics, with biophony being highest in grazed forests and lowest in ungrazed forests in winter. Livestock shifted the forest soundscape composition by increasing the audibility of birds and insects while decreasing the vocalizations of sika deer (Cervus nippon) and crows, resulting in reduced sound diversity and complexity in grazed forests. We also found that grazing can reduce the leaf area index, herbaceous plants, and canopy density, which can influence these effects indirectly. Interestingly, cowbells noticeably altered the dawn chorus of birds; during spring and summer grazing periods, the chorus was characterized by an increased bird calling rate and greater vocal complexity (elevated Acoustic Complexity Index), patterns consistent with a behavioral adjustment to acoustic masking. This study highlights how livestock modify forest acoustic communities. To preserve natural soundscapes, we suggest mitigating cowbell noise through silent trackers (e.g., GPS) or reduced bell density in priority zones. Sustainable practices, including rotational grazing and buffer zones, are also vital to maintain forest structure and acoustic diversity. We suggest that integrating SED models with acoustic indices provides a robust framework for monitoring such anthropogenic disturbances.

PMID 42503024
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PubMedMobile DNA2026-07-16

Transposable element dynamics and regulatory role in sika deer (Cervus nippon) antler development.

Wang Qianghui Q, Xing Haihua H, Ma Yukai Y, Sun Zihui Z et al.

Deer antlers represent one of the few mammalian organs capable of complete regeneration, yet the underlying genomic regulatory mechanisms remain incompletely understood. Transposable elements (TEs), as key drivers of genome evolution and gene regulation, may play pivotal roles in the evolution of complex traits. This study aimed to systematically investigate the evolutionary dynamics of TEs in sika deer genome and to elucidate their potential regulatory functions in the development of antler by integrating comparative and functional genomics approaches. Comparative genomics revealed a lineage-specific massive expansion of LINE retrotransposons (dominated by RTE-BovB and L1 subfamilies) in cervid genomes, particularly in sika deer and red deer, where they constitute over 29% of the genomic sequence. The peak of this expansion (~ 7.5 million years ago) coincides with the major cladogenesis events within Cervus. Expression analysis showed that approximately 8.88% of annotated TEs are transcriptionally active in antler mesenchyme, with LINE and LTR elements being predominant among the 1,191 TEs consistently highly expressed across all stages. We identified numerous stage-specifically expressed TEs (SETEs) and found positive correlations between SETEs and key antler development genes, such as the osteogenic master regulator RUNX2, the extracellular matrix remodeling gene ANPEP, and the collagen synthesis gene P4HA3. Enrichment analysis demonstrated that genes adjacent to these TEs are significantly involved in pathways crucial for regeneration and rapid growth, including Wnt signaling, Hippo signaling, regulation of the actin cytoskeleton, and protein digestion and absorption. Our findings point to a potential role for cervid TEs expansion in driving genomic evolution and the acquisition of cervid-specific phenotypes, particularly antler growth and development. Through profiling TE expression in antler mesenchymal tissue across key development stages, the results suggest that dynamic TEs expression may be involved in the regulation of antler development, implicating a potential regulatory role for TEs in this rapid growth process. This study provides new insights into the molecular mechanisms underlying the rapid growth of antlers.

PMID 42458577
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PubMedInternational journal of gynaecology and obstetrics: the official organ of the International Federation of Gynaecology and Obstetrics2026-07-15

Assessment and management of dyspareunia in peri- and postmenopausal women: A phenotype-based gynecologic approach.

Broul Marek M, Vančo Marcel M, Banýrová Jaroslava J, Hujová Aneta A

Dyspareunia in peri- and postmenopausal women is common, clinically consequential, and often undertreated in gynecologic practice. Although genitourinary syndrome of menopause (GSM) is a frequent contributor, intercourse-related pain may also reflect vestibular, pelvic floor, dermatologic, inflammatory, treatment-related, and psychosocial factors. This narrative review provides a practical phenotype-based framework for assessment and management when GSM, vestibular pain, and pelvic floor dysfunction coexist, and when deep-pain phenotypes require broader pelvic evaluation. PubMed/MEDLINE, the Cochrane Library, and selected guideline sources were searched for English-language literature published from January 2014 to March 2026, prioritizing guidelines, systematic reviews, randomized or sham-controlled trials, and examination-based studies relevant to office gynecology. History should distinguish superficial from deep pain, provoked from spontaneous symptoms, and urinary, dermatologic, inflammatory, and psychosocial features. Examination should proceed from vulva and vestibule to vagina and pelvic floor, with bimanual assessment and selective imaging when deeper pathology is suspected. Management includes education, irritant avoidance, moisturizers and lubricants, and prescription therapy for clinically significant GSM, usually low-dose vaginal estrogen, with prasterone or ospemifene as selected alternatives. Pelvic floor physiotherapy should be considered when tenderness, guarding, or penetration-limiting hypertonicity is present. Because menopause-specific pelvic floor evidence remains limited, related recommendations are framed as cautious extrapolations from broader dyspareunia, vulvodynia, and chronic pelvic pain literature.

PMID 42454524
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PubMedInternational journal for parasitology. Parasites and wildlife2026-07-13

Phylogenetic and molecular insights into the genetic diversity of the invasive nematode Ashworthius sidemi infecting Poland's free-ranging European bison (Bison bonasus).

Świsłocka-Cutter Magdalena M, Borkowska Anetta A, Kowalczyk Rafał R, Kołodziej-Sobocińska Marta M

The invasive blood-sucking nematode Ashworthius sidemi, originally parasitising Asian cervids, has spread across Europe following human-mediated introductions of sika deer (Cervus nippon). In this study, we characterised the molecular variation of A. sidemi obtained from two neighbouring populations of European bison (Bison bonasus) in northeastern Poland, located in the Białowieża Primeval Forest and Knyszyńska Forest. Individual worms (one per host) were analysed using nuclear molecular markers (18S rRNA, 28S rRNA, ITS-1) and mitochondrial markers (COX1, ND4). All analysed markers revealed no detectable intraspecific genetic variability among the 16 specimens sequenced, with a single haplotype identified for each marker. This finding is consistent with a founder effect and/or recent introduction of the parasite. The genetic homogeneity observed across geographically close bison herds may also reflect host mobility. Phylogenetic analyses based on both nuclear and mitochondrial markers consistently placed A. sidemi within the subfamily Haemonchinae, closely related to Haemonchus spp. and Mecistocirrus digitatus. The ITS-1, COX1, and ND4 markers provided sufficient resolution to differentiate A. sidemi from other Trichostrongylidae species, whereas the 18S and 28S rRNA genes were too conserved to discriminate species- or subfamily-level relationships. Our findings demonstrate the utility of nuclear and mitochondrial markers for the identification and phylogenetic classification of trichostrongyloid nematodes. These results provide important insights into the invasion dynamics of A. sidemi, which may support parasite surveillance and conservation efforts of endangered host species.

PMID 42438769
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PubMedAnimal science journal = Nihon chikusan Gakkaiho2026-07-11

Diversity of the Major Histocompatibility Complex Region Among Seven Founders of the Crested Ibis Nipponia nippon in Japan.

Taniguchi Yukio Y, Yamada Takahisa T, Sugiyama Toshie T, Kaneko Yoshinori Y et al.

The Crested Ibis Nipponia nippon is a critically threatened avian species. The current Japanese population originates from only seven founders introduced from China. The major histocompatibility complex (MHC) is a highly polymorphic genomic region that plays a central role in the immune system. We previously reported that only three MHC class II haplotypes (HP1-3) with one to three copies of MHC-IIA/IIB gene pairs (one copy of DAA/DAB locus and 0-2 copies of DBA/DBB loci) were detected among the five older founders, and four MHC-IIB exon 2 alleles (Type I-IV) were identified. In this study, MHC class II haplotypes in two novel founders, and MHC class IA genotypes at UAA locus in the seven founders were investigated. Of the two novel founders, while one possessed known HP1 and HP2, another possessed known HP1 and a novel haplotype (HP4) with the combination of type II and type I in DAB and DBB exon 2 s, respectively. Analysis of the linkage between MHC class II haplotypes and UAA alleles revealed five distinct MHC haplotypes against seven founders. These results strongly suggested that the founders might be considerably closely related, and the novel HP4 was produced by recombination between HP1 and HP2.

PMID 42433167
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