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Fraction F (Fraction F / Ateroid / Ateroid 200)

✓ Approved

Gentium · 治疗药物

什么是 Fraction F?

Fraction F 是一种治疗药物,由Gentium研发。该药已获批,用于治疗相关适应症,给药途径:Injectable (Others)、Intravenous (IV)、Oral (PO)。

药物档案

商品名Fraction F, Ateroid, Ateroid 200
公司Gentium
给药途径Injectable (Others), Intravenous (IV), Oral (PO)
状态Approved

治疗适应症

Fraction F 针对 1 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Nervous system disordersDementia Alzheimer's type✓ Approved

相关研究文献

PubMedBiophotonics discovery2026-09-10

Transient infrared laser exposure modulates calcium activity in cortical dendritic spines.

Hardenburger Jacob J, Grow George G, Rasiah Pratheepa P, Gerges Mona M et al.

Infrared neural stimulation (INS) is an optical neuromodulation technique that elicits neural activity through photothermal temperature gradients. Photothermal gradients have been shown to alter neuronal excitability, but the effects on the dendritic spine (DS) structure and function have not been characterized. We aim to determine whether INS induces calcium signaling in DS and whether this signaling alters filamentous actin (F-actin). We used confocal imaging of cortical neurons expressing a genetically encoded calcium indicator (GCaMP)8f-Syn1 and mCardinal-LifeAct during laser exposure. Fluorescence signals were measured within regions of interest covering the DS. The resulting fluorescence measurements were baseline-normalized, and transient spiking activity in DS was quantified. Transient thermal gradients induce persistent calcium activity in a fraction of DS, independent of pulse duration but dependent on the absolute temperature and number of laser exposures. There is no relationship between the calcium activity and F-actin. Calcium signaling in DS was not mediated by ionotropic glutamate receptors but depended on extracellular entry. These results indicate that transient thermal gradients elicit calcium activity in DS, but the induced activity does not alter F-actin, suggesting that transient thermal gradients may be a useful tool for studying calcium dynamics in DS without triggering traditional structural plasticity pathways.

PMID 42719458
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PubMedChemistry & biodiversity2026-09-10

Antioxidant Activities of Pentacyclic Triterpenes From Melipona beecheii Propolis and Their Semisynthetic Derivatives.

Santana-Hernández Aarón A, Yam-Puc Alejandro A, Yah-Nahuat Pamela P, Vargas-Vargas María M et al.

Four principal fractions (I-IV) were obtained from the Melipona beecheii propolis. GC-MS analysis of these fractions allowed us to recognize 11 pentacyclic triterpenes (PTs), fraction I [β-amyrin acetate (1), germanicol acetate (2), moretenol acetate (3) and 24-methylencycloartan-3-ol acetate (4)]; fraction II [marsformosanone (5), β-amyrenone (6), germanicone (7) and lupenone (8)]; fraction III [β-amyrin (9) and, glutinol (10)]; and fraction IV [9 and α-amyrin (11)]. This is the first time that triterpenes 7 and 10 are reported in the propolis of M. beecheii. Three semisynthetic derivatives were prepared: the reduction of fraction II and the acetylation and oxidation of fraction IV. The ethanolic extract of propolis and fraction III presented the highest free DPPH radical scavenging capacity at 53.89 ± 8.39% and 47.77 ± 0.91%, respectively, using a concentration of 10 mg/mL. In contrast, the reducing power of Fe (III) analysis showed a strong reducing power of Fe(III) for all fractions and their derivatives with an EC50 = 0.8-1.0 mg/mL.

PMID 42720076
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PubMedJAC-antimicrobial resistance2026-09-10

Performance of the Sensititre YeastOne assay compared with EUCAST E.Def 9.4 against Fusarium clinical isolates: focus on voriconazole and amphotericin B.

Chen Pao-Yu PY, Wu Un-In UI, Liu Wang-Da WD, Huang Yu-Tsung YT et al.

Despite the global emergence of Fusarium infections, data validating commercial antifungal susceptibility testing against these moulds remain scarce. We evaluated the performance and optimal reading time of the Sensititre YeastOne (SYO) assay against Fusarium clinical isolates compared with the EUCAST reference method. This two-centre study (2011-2023) analysed 123 Fusarium isolates identified via two-step molecular sequencing. In vitro susceptibilities to voriconazole and amphotericin B were evaluated using SYO (24 h and 48 h readouts) versus the EUCAST E.Def 9.4 broth microdilution reference method (48 h readout). Essential agreement (EA) was defined as a ±2 log2 dilution difference; >90% was acceptable. Fusarium solani species complex (FSSC) dominated the cohort (85.3%), predominantly F. keratoplasticum and F. pseudensiforme. EUCAST testing revealed high MIC50/MIC90 values of voriconazole (>16/>16 mg/L) and amphotericin B (2/16 mg/L). While 65% (80/123) of isolates displayed positivity by SYO at 24 h, median spectrophotometric growth was significantly greater at 48 h than at 24 h [0.37 (IQR 0.315-0.403) versus 0.18 (0.151-0.206)]. At 48 h, EA approached acceptability for voriconazole (92.7%) and amphotericin B (89.4%). Voriconazole categorical agreement (CA) among FSSC was 88.6% and reached 96.9% for F. pseudensiforme. For amphotericin B, SYO MICs clustered around 4-8 mg/L, yielding 100% very major error for F. keratoplasticum and F. pseudensiforme but 100% CA for F. falciforme, F. petroliphilum and non-FSSC. Voriconazole and amphotericin B susceptibility determined by SYO cannot universally replace reference methods due to failure to detect non-WT to amphotericin B for prevalent species within FSSC. However, alongside accurate species-level molecular identification, SYO provides actionable susceptibility data for validated species-antifungal combinations.

PMID 42718997
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PubMedFrontiers in cellular and infection microbiology2026-09-10

NS2A V89F mutation in a DENV1 clinical isolate enhances neurotropism and neuroinvasion.

Zhao Yuqi Y, Wang Linqing L, Lin Yifan Y, Chen Yangyang Y et al.

Dengue virus (DENV) neurological complications are increasingly reported, yet the viral genetic determinants of neurotropism remain poorly characterized. We screened 25 DENV1 clinical isolates from the 2014 outbreak in Guangdong, China, for neurotropism in suckling mice, and integrated comparative genomics, pre-expression functional assays, population-scale sequence analysis, and OpenFold3 structural modeling to identify mutations associated with enhanced neuroinvasion. We found that only strain P1253 induced neurological symptoms and mortality via subcutaneous inoculation, producing cortical-selective lesions distinct from the diffuse encephalitic damage observed after intracranial inoculation, and P1253 replicated preferentially in human brain microvascular endothelial cells (HBMEC) compared to contemporaneous strains. Comparative genomics identified three unique mutations in P1253 (NS1 175Y→H, NS2A 89V→F, NS4A 2V→I), and pre-expression assays demonstrated that only NS2A 89V→F significantly enhanced viral replication and cytopathic effect in HBMEC. Analysis of 1,990 complete DENV1 genomes revealed five natural mutant types in the NS2A 89 -96 residue region, with P1253 representing the FIPI quadruple-mutant type, and OpenFold3 structural prediction showed that 89V→F introduced on the VIPI background induced the most significant distal domain reorientation (RMSD 1.605 Å), increasing the centroid-to-centroid distance between residues 89 -96 and 185 -218 from 18.221 Å to 27.462 Å. These findings identify NS2A 89V→F as a candidate adaptive mutation associated with enhanced neurotropism in DENV1 and provide a framework for monitoring neurovirulent variants.

PMID 42718655
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PubMedCardiovascular diagnosis and therapy2026-09-10

Statistical concerns regarding the validation of myocardial contraction fraction cut-off in transcatheter aortic valve replacement patients.

Coskun Senol S

PMID 42719204
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PubMedBiopolymers2026-09-10

Pre-Esterification Dry Heat Treatment Enhances the Functional Properties of Starch Citrate: Enzyme Resistance and Water Absorption.

Dogadina Anna A, Tryakhov Denis D, Grishkova Svetlana S, Maslennikov Daniel D

This study investigates how pre-esterification dry heat treatment (DHT) of corn starch at 170°C, 180°C, and 200°C influences the functional properties of subsequently synthesized starch citrates. Structural and morphological changes induced by DHT and esterification were analyzed using scanning electron microscopy, X-ray diffractometry, and Fourier-Transform Infrared spectroscopy. Starch citrates were characterized for their resistance to pancreatic α-amylase and amyloglucosidase, as well as their water absorption capacity (WAC) at 37°C. Results demonstrated a strong correlation between DHT temperature and the functional properties of the final citrate. Increasing the DHT temperature significantly increased the resistant starch fraction and WAC. Specifically, citrates from native starch had a resistant starch (RS) fraction of 91%, while citrates from starch pre-treated at 200°C exhibited a markedly increased RS fraction of 98% and a 64% increase in WAC. These findings indicate that DHT is an effective pre-treatment for enhancing the dietary fiber potential and hydration properties of starch citrates.

PMID 42717628
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